In Vitro Antiplasmodial Activity of Sesquiterpene Lactones from Ambrosia tenuifolia

المؤلفون المشاركون

Giménez-Turba, Alberto
Sülsen, Valeria P.
Martino, Virginia S.
Muschietti, Liliana V.
Laurella, Laura C.
Anesini, Claudia
Gutierrez Yappu, D.

المصدر

Evidence-Based Complementary and Alternative Medicine

العدد

المجلد 2011، العدد 2011 (31 ديسمبر/كانون الأول 2011)، ص ص. 1-4، 4ص.

الناشر

Hindawi Publishing Corporation

تاريخ النشر

2011-05-25

دولة النشر

مصر

عدد الصفحات

4

التخصصات الرئيسية

الطب البشري

الملخص EN

The in vitro antiplasmodial activity of Ambrosia tenuifolia organic extract and its isolated sesquiterpene lactones, psilostachyin and peruvin, has been evaluated against Plasmodium falciparum F32 and W2 strains.

The cytotoxicity of both compounds was determined on lymphoid cells, and their corresponding selectivity indexes (SIs) were calculated.

Peruvin was the most active compound on F32 strain of P.

falciparum with a 50% inhibitory concentration value (IC50) of 0.3 μg/mL (1.1 μM) whereas psilostachyin showed activity on both strains (IC50 = 0.6 (2.1 μM) and 1.8 μg/mL (6.4 μM)).

Fifty percent cytotoxic concentration (CC50) values (48 h) were 6.8 μg/mL (24.3 μM) and 10.0 μg/mL (37.9 μM) for psilostachyin and peruvin, respectively.

نمط استشهاد جمعية علماء النفس الأمريكية (APA)

Sülsen, Valeria P.& Gutierrez Yappu, D.& Laurella, Laura C.& Anesini, Claudia& Giménez-Turba, Alberto& Martino, Virginia S.…[et al.]. 2011. In Vitro Antiplasmodial Activity of Sesquiterpene Lactones from Ambrosia tenuifolia. Evidence-Based Complementary and Alternative Medicine،Vol. 2011, no. 2011, pp.1-4.
https://search.emarefa.net/detail/BIM-465184

نمط استشهاد الجمعية الأمريكية للغات الحديثة (MLA)

Sülsen, Valeria P.…[et al.]. In Vitro Antiplasmodial Activity of Sesquiterpene Lactones from Ambrosia tenuifolia. Evidence-Based Complementary and Alternative Medicine No. 2011 (2011), pp.1-4.
https://search.emarefa.net/detail/BIM-465184

نمط استشهاد الجمعية الطبية الأمريكية (AMA)

Sülsen, Valeria P.& Gutierrez Yappu, D.& Laurella, Laura C.& Anesini, Claudia& Giménez-Turba, Alberto& Martino, Virginia S.…[et al.]. In Vitro Antiplasmodial Activity of Sesquiterpene Lactones from Ambrosia tenuifolia. Evidence-Based Complementary and Alternative Medicine. 2011. Vol. 2011, no. 2011, pp.1-4.
https://search.emarefa.net/detail/BIM-465184

نوع البيانات

مقالات

لغة النص

الإنجليزية

الملاحظات

Includes bibliographical references

رقم السجل

BIM-465184